Heme degradation

 

Heme Degradation: From Heme to Bilirubin

Heme from senescent red blood cells is degraded primarily in the reticuloendothelial system (spleen and liver).

Step Enzyme/Process Key Transformation
Step 1 Heme Oxygenase Opens the heme ring to produce biliverdin (green pigment), CO, and Fe2+.
Step 2 Biliverdin Reductase Reduces biliverdin to unconjugated bilirubin (yellow pigment).
Transport Albumin Unconjugated bilirubin is insoluble; it travels bound to albumin to the liver.
Conjugation UDP-glucuronosyltransferase Conjugates bilirubin with glucuronic acid to increase water solubility.
High-Yield Core Realities:

  • Unconjugated vs. Conjugated: Unconjugated bilirubin is toxic (lipid-soluble) and can cause kernicterus in neonates. Conjugated bilirubin is non-toxic and water-soluble, excreted into bile.
  • Clinical Significance: Elevated unconjugated bilirubin suggests pre-hepatic (hemolysis) or hepatic causes (Gilbert syndrome). Elevated conjugated bilirubin suggests obstructive (biliary) or hepatobiliary pathology.
  • Enterohepatic Cycling: Bacteria in the intestine convert conjugated bilirubin into urobilinogen, which is either excreted in feces as stercobilin or reabsorbed and excreted in urine as urobilin.